ID Refrence Source Clone name Sequence Motif Target-tumor Target-cell Receptors-biomarker Phage/Library In vitro/Ex-vivo In vivo Homing/targeting Payloads Patent
1001He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R22CSNIDARACNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cells, H460 CellBALB/ C mice with lung tumorHomingLiposomal doxorubicinUS2010/0233161A1
1002He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.3R5CDPSRGKNCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1003He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R24CPSDLKDACNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1004He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R4CRTTRGTKCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1005He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R8CRMTRNKPCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1006He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R17CRVSRQNKCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1007He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.4R9CAKIDPELCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1008He X et al. Mol Pharm. 2011 Apr 4;8(2):430-8.3R14CGGERGKSCNALung (major), Colon, Breast cancerTumor cellNAT7 phage / CX7C peptide libraryH460, A549 cells, H226 cells, SNU484, MDA-MB-231, HT29 cellsNATargetingNAUS2010/0233161A1
1116Jiang YQ et al. Mol Med. 2006 Apr-Jun;12(4-6):81-7.HCC79KSLSRHDHIHHHNAHepatocellular carcinomaTumor cellHer-2 and ErbB-2M13/ 12-mer peptide libraryHuman hepatoma cell line SMMC-7721, BEL-7402, and HL-02BABL/c mice HomingToxic shock syndrome toxin 1 (TSST-1)US 2009/0274625 A1
1127Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANRLKCRAQATHSAAPCIRGYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1128Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NARQNSCTYSDARRWALCWSGENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1129Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAQLNSCIHSGDRAIRGCMDWVNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1130Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAKYGLCRDETVFPSHSCTFTGNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1131Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGSPQCPGGFNCPRCDCGAGYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1132Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGTGSCGYGKLHTGYWCSYFPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1133Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANSSSCDTSVVRSTWACILQPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1134Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVRAVCTTLKSRGHEECWSLQNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1135Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVYAQCGVNVRTGRGGCSRLMNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1136Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAVHMNCSWMRVSEGHPCESADNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1137Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGRQGCYEHLWRLIAWCAIFLNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1138Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NALRMTCAFGVAQRSADCALSSNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1139Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NASIVNCSAALTDLPTRCGGNINABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1140Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NACGTRCVRCQNGPEASCEQPLNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1141Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NATPLFCGNHGRQPSPLCMKWDNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1142Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAFTTVCRQPRGHEAIVCGSGKNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1143Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAAPSFCGTAMLGASRYCYSGPNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1144Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGARECESGGPGMRKLCTQINNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1145Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NANNRACFRTSKGNPAECPYLGNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1146Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAGSLACQNIVVCVKKQCNALCNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1147Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NAKRASCQNPLFSNFFVCGLSENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1148Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NALPNFCMDTSGRAGPLCMGSENABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1149Krag DN et al. Cancer Res. 2006 Aug 1;66(15):7724-33.NARHTVCRVSLSSVQGSCSHEYNABreast cancerTumor cellNAM13 phage/Random 20 mer (X4CX10CX4) peptide libraryPatient biopsies, cancer cell line (breast: SK-BR-3), T47D, BT474, MDA-MB-231 and MDA-MB-361NAHoming (Phage display clone)NANA
1152Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.peptide 20GRRTRSRRLRRSNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHomingNANA
1153Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 1, 3, 6SMSIASPQIPWSNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1154Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 2, 4, 10, 23TPRNLRTSNTHRNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1155Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 5, 11, 15, 19, 25GRRIAGPYIALENAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1156Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 7, 9, 13, 18SMPINSPYIPWSNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1157Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 8, 16GRRPMKLNKTPNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1158Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 12, 14, 17GRRINRLILPRNNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1159Hu S et al. Biochem Biophys Res Commun. 2006 Mar 24;341(4):964-72.Phage 27, 28GRRTRSSRLRNSNAGastric cancer, Liver metastassisTumor cellNAM13PIII phage/12 mer random peptide libraryHuman gastric cancer cell line XGC9811, XGC9811(liver metastatic gastric cell line) LAGS, MKN45BALB/c nude mice( 4- to 5-weeks-old) bearing human gastric carcinoma cell line XGC9811 xenograftHoming (Phage display clone)NANA
1166Zurita AJ et al. Cancer Res. 2004 Jan 15;64(2):435-9.NACGRRAGGSCNAProstate cancerTumor cellIL-11 receptorNAHuman primary and metastatic prostate cancer samples,cancer-derived cell lines MDA-PCa-2b and LNCaPNATargetingNAWO0402020722A2
1169Kondo M et al. Int J Cancer. 2004 Jan 10;108(2):301-6.GPLPLR-Lip. DPP-CNDAC peptideGPLPLRPLPTumor metastasisAngiogenic endothelium cell,tumor cell.MT1-MMP(Membrane type 1Matrix metalloproteinase )NANA5-week-old BALB/c male mice bearing NL-17 carcinoma HomingRibosome-encapsulated [2-18F]FDG,Lip. DPP-CNDAC peptideNA
1192Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.RPMrel peptide CPIEDRPMCNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29, Human biopsiesNATargetingMtochondrial toxin (KLAKLAK)2US 7,452,965b2
1193Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAPIEDRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1194Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAPIDERPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1195Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAALRDRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1196Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAPMMRQRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1197Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAPLASRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1198Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAPEKFRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1199Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAVPEQRPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1200Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NADLPMHPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1201Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAQFQSQPMNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1202Kelly KA et al. Neoplasia. 2003 Sep-Oct;5(5):437-44.NAQPPMEYSNAColorectal cancerTumor cellNAM13 phage/ CX7C peptide libraryColon carcinoma cells (HT29), well-differentiated colon carcinoma cells (HCT116), HT29NATargetingNANA
1219Shadidi M et al. FASEB J. 2003 Feb;17(2):256-8.GFP-peptide fusion proteinsLTVSPWYNABreast cancerTumor cellErbB2M13 phage/7 mer peptide libraryThe breast cancer cell lines SK-BR-3, T47D, PM1,HT2933.NATargetingGFPNA
1220Shadidi M et al. FASEB J. 2003 Feb;17(2):256-8.NATLTVLPWNABreast cancerTumor cellErbB2M13 phage/7 mer peptide libraryThe breast cancer cell lines SK-BR-3NATargetingNANA
1221Shadidi M et al. FASEB J. 2003 Feb;17(2):256-8.NANLYVASWNABreast cancerTumor cellErbB2M13 phage/7 mer peptide libraryThe breast cancer cell lines SK-BR-3NATargetingNANA
1238Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMARSGLNAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR3NATargeting & further studiedNANA
1239Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMARAKENAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR4NATargeting & further studiedNANA
1240Houimel M et al. Int J Cancer. 2001 Jun 1;92(5):748-55.NAMSRTMSNAHuman breast and ovarian adenocarcinomasTumor cellErbB-2NASK-BR-3, MDA-MB-468, OVCAR5NATargeting & further studiedNANA
1251Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1.1AEGEFMYWGDSHWLQYWYEGDPAKNABreast cancerTumor cellErbB-2T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1252Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1AEGEFWGDSHWLQYWYEGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1253Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL2AEGEFIHNRYNRFFYWYGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1254Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1.2AEGEFPRWGDSHWLQYWYEGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1255Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1.3AEGEFLMWGGSHWLEYWYEGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1256Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1.4AEGEFGHWCDQHWLQYWYEGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1257Urbanelli L et al. J Mol Biol. 2001 Nov 9;313(5):965-76.NL1.5AEGEFGWWGDSHWLQYEGDPAKNABreast cancerTumor cellHER2(Human epidermal growth factor receptor 2) T7 phage/12 mer peptide libraryHuman breast carcinoma SK-Br-3, human ovarian carcinoma SKOV3, human melanoma MeWo and mouse fibroblast NIH3T3 cellsNATargetingNANA
1258Aoki Y et al. Cancer Gene Ther. 2001 Oct;8(10):783-7.NACRGDCFRGDHepatic and pancreatic cancerTumor cellIntegrinsNAHuman hepatoma cell lines ( PLC / PRF / 5 andHepG2 ) ,human pancreatic cancer cell lines ( Hs700T and MIAPaCa - 2 )Male BALB /c mice HomingHistidylated oligolysine plasmid , bafliomycinNA
1259Aoki Y et al. Cancer Gene Ther. 2001 Oct;8(10):783-7.NACDCRGDCFCRGDHepatic and pancreatic cancerTumor cellIntegrinsNAHuman hepatoma cell lines ( PLC / PRF / 5 andHepG2 ) ,human pancreatic cancer cell lines ( Hs700T and MIAPaCa - 2 )NATargetingNAUS 2003/0152578 A1
1260Aoki Y et al. Cancer Gene Ther. 2001 Oct;8(10):783-7.NACNGRCVSGCAGRCNGRHepatic and pancreatic cancerTumor cellIntegrinsNAHuman hepatoma cell lines ( PLC / PRF / 5 andHepG2 ) ,human pancreatic cancer cell lines ( Hs700T and MIAPaCa - 2 )NATargetingNAWO06067633A2
1261NANACGSLVRCGSLBreast tumorTumor cellNAPhagedisplaying an Arg ­ Gly ­ Asp ( RGD ) ­ containing peptideNAMice bearing human 435 breast carcinomaHomingDoxorubicinUS 2003/0152578 A1
1262Chen Y et al. Cancer Res. 2001 Mar 15;61(6):2434-8.NACRGDCGGKWCFRVCYRGICYRRCRRGDProstate cancer, MelanomaTumor cell and Endothelial cellIntegrinsNAThe TSU human prostate cancer cells, B16 melanoma, nontumorigenic cell lines Cos-7, and NIH-3T3CAMs of 10-day-old chicken embryos, C57BL/6 mice bearing B16 melanoma HomingAntimicrobial peptideNA
1263Spear MA et al. Cancer Gene Ther. 2001 Jul;8(7):506-11.NAMCPKHPLGCNAMalignant gliomasTumor cellNACMTI phage /30 mer peptide libraryU87 - MG human malignant glioma , T98 - MG human malignant glioma , ,AST- 4 human malignant glioma,PANC - 1 humanpancreatic adenocarcinoma , 9L rat malignant glioma cellsNATargetingNANA
1264Spear MA et al. Cancer Gene Ther. 2001 Jul;8(7):506-11.NALCPKHPLGCNAMalignant gliomasTumor cellNACMTI phage /30 mer peptide libraryU87 - MG human malignant glioma , T98 - MG human malignant glioma , ,AST- 4 human malignant glioma,PANC - 1 humanpancreatic adenocarcinoma , 9L rat malignant glioma cellsNATargetingNANA
1293Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NATAASGVRSMHNAMelanomaTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NG2 knockout mice, NG2 expressing wild mice.HomingNAUS 6,528,481 B1
1294Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NALTLRWVGLMSNAMelanomaTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NG2 knockout mice, NG2 expressing wild mice.HomingNAUS 6,528,481 B1
1295Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAGGGTRAGMKYNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1296Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAWGKIEDPLRANATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1297Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAAGQTLTASGDNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1298Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NADLLAVSWLRANATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1299Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NASAERGVVAMSNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1300Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAAIHSELMWVSNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1301Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAFWTERAGWAYNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1302Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAMVWSKGPLFLNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1303Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAAGTRMSWEVLNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1304Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAVSRSSRWGSINATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1305Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NADAHVLVPRTPNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1306Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NAAQGIVLQLALNATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1307Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NALSPLLSPATANATumor neovasculatureTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NATargetingNAUS 6,528,481 B1
1320Drecoll E et al. PLoS One. 2009 May 27;4(5):e5715.F3KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKNAPeritoneal carcinomatosisNucleus of tumor cellsNucleoinNAEMT6, MIAPACA, CMT93, OVCAR3, MDA-MB-435 cell lineMice bearing intra-peritoneal MDA-MB-435 xenograft tumorsHomingBi-DTPA-[F3]2EP1783140A3,US 7,544,767B2
1323Karmali PP et al. Nanomedicine. 2009 Mar;5(1):73-82.LyP-1CGQKRTRGCNABreast cancerTumor lymphatics, Tumor cellsp32 and gC1gRNANAMice bearing MDA-MB-435 human cancer xenograftsHomingQuantum dotsUS 2010/0172 835 A1
1328Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDKGPDCRGDProstate, Pancreatic ductal, breast cancer, bone , brain, cervical cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNude mice with multiple tumors (prostrate PC-3, PPC1, 22RVI Xenograft), (pancreatic MIAPaCa-2 Xenograft)HomingIron oxide nanoworms, iRGD-linked abraxaneUS 2009/0246133A1
1329Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDRGPDCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNANA
1330Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDKTTNCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNANA
1331Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDHAGDCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNANA
1332Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDHGVECRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1333Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACGRGDNLPCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1334Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACGRGDNLACRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1335Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACEKRGDNLCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1336Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACEKRGDSVCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1337Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACSGRGDSLCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1338Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACGKRGDSICRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1339Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACTGRGDALCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1340Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDSACRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1341Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDKGENCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1342Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACGRGDSPDCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1343Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDKGPECRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1344Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDKHADCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1345Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDHAANCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1346Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACRGDAGINCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1347Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACGRGDMPSCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1348Sugahara KN et al. Cancer Cell. 2009 Dec 8;16(6):510-20.NACEKRGDSLCRGDProstate cancerEndothelial cell and tumor cellAlpha 5 beta 3 and Alpha 5 beta 5 integrins neuropilin-1T7 phage / CX7C peptide libraryCultured PPC1 human prostate cancer cells, M21 human melanoma cellsNATargetingNAUS 2009/0246133A1
1349Park JH et al. Small. 2009 Mar;5(6):694-700.F3KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKNABreast cancer ,FibrosarcomaEndothelial cell and tumor cellNANANAMice bearing human (MDA-MB-435 human carcinoma and HT1080 human fibrosarcoma) xenograftHomingSuperparamagnetic nanospheres, superparamagnetic IO nanoworms (NWs)US 7,544,767 B2
1372Huang EH et al. J Surg Res. 2009 Aug;155(2):231-6.CTCE-9908KGVSLSYRKKGVSLSYRNABreast cancerTumor cellCXCR4 receptorNAMDA-231humanbreast adenocarcinoma cell line , MDA-231-BSC-12Female athymic nude mice (4-6 weeks)HomingFITCNA
1387Kumar SR et al. Clin Cancer Res. 2007 Oct 15;13(20):6070-9.NAKCCYSLNAHuman breast carcinomaTumor cellErbB-2NAMDA-MB,Human breast carcinoma cell line, Prostate carcinoma cell line (PC-3),K-562 human erythroid leukemia cell lineSCID mice, MDA-MB-435 breast carcinoma cellHoming111In-DOTA, BiotinUS 2010/0061930
1390Zhang B et al. Mol Med. 2007 May-Jun;13(5-6):246-54.Synthetic peptide HCBP1FQHPSFINAHepatoma cancerTumor cellNAM13 phage /7- mer peptide libraryHepatocellular carcinoma cell line (HepG2),Hepatocellular carcinoma cell line (HepG2),Normal hepatocyte line (L-02) ,The hepatocellular carcinoma cell lines and BEL-7402, Passage cell line of human cervical cancer Hela,Human patients biopsiesBalb-c mice bearing HepG2 xenograftsHomingFITCNA
1454Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-A9PQNSKIPGPTFLDPHP-(C)-G-P-XXX-D(C)-PTumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549 trans, Human breast carcinoma cell line MDA-MB-435, Human prostate carcinoma cell line PC-3M, MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1455Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A3SMEPALPDWWWKMFKNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 3NATargetingNANA
1456Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A4DKPTAFVSVYLKTALNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 4NATargetingNANA
1457Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A18APRPGPWLWSNADSVNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 5NATargetingNANA
1458Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A19GVTDSSTSNLDMPHWNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 6NATargetingNANA
1459Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A28PKMTLQRSNIRPSMPNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 7NATargetingNANA
1460Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-A40LYPLHTYTPLSLPLFNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 8NATargetingNANA
1461Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-C4LTGTCLQYQSRCGNTRNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans express galactein 9NATargetingNANA
1462Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-C9AYTKCSRQWRTCMTTHNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3M,MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1463Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.G3-C12ANTPCGPYTHDCPVKRP-(C)-G-P-XXX-D(C)-PTumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide libraryHuman breast cancer cell lines BT549, express detectable levels of galectin-3, BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3M,MDA-MB-435 human breast carcinoma cells on HBME-1 monolayersNATargeting & further studiedNANA
1464Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-C44NISRCTHPFMACGKQSNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide librarySaos2 (derived from a human osteosarcoma),Human breast cancer cell lines BT549, express detectable levels of galectin-3 ,BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3MNATargetingNANA
1465Zou J et al. Carcinogenesis. 2005 Feb;26(2):309-18.Clone G3-C60PRNICSRRDPTCWTTYNATumor metastasisEndothelial cell and tumor cellGalectin-3f88 phage/15mer peptide library and f88 phage/Cys6 mer peptide librarySaos2 (derived from a human osteosarcoma),Human breast cancer cell lines BT549, express detectable levels of galectin-3 ,BT549trans,Human breast carcinoma cell line MDA-MB-435,Human prostate carcinoma cell line PC-3MNATargetingNANA
1473Askoxylakis V et al. Clin Cancer Res. 2005 Sep 15;11(18):6705-12.p160VPWMEPAYQRFLNAHuman breast cancerTumor cellNANABreast cancer cell line MDA-MB-435,neuroblastoma cell line WAC 2, MCF-7Female BALB/c nu/nu mice carrying human breast cancer MDA-MB-435 tumorsHoming(131)I-labeled and the FITC-labeledNA
1474Funovics M et al. Neoplasia. 2005 Oct;7(10):904-11.NABCDSDSDITWDQLWDLMKNAHuman prostrate cancer, lewis lung carcinomaTumor cell,endothelial cellE-selectinNAActivated HUVEC, Human prostrate biopsies,llc cell lineMouse xenograft model of LLCHomingFITC , nanoparticle CLIO(Cy5.5)NA